Lack of Interaction Between the Peptidomimetic Substrates Captopril and Cephradine
dc.contributor.author | Foster, David R. | en_US |
dc.contributor.author | Yee, Shiyin | en_US |
dc.contributor.author | Bleske, Barry E. | en_US |
dc.contributor.author | Carver, Peggy L. | en_US |
dc.contributor.author | Shea, Michael J. | en_US |
dc.contributor.author | Menon, Sujatha S. | en_US |
dc.contributor.author | Ramachandran, Chandrasekharan | en_US |
dc.contributor.author | Welage, Lynda S. | en_US |
dc.contributor.author | Amidon, Gordon L. | en_US |
dc.date.accessioned | 2013-04-08T20:50:00Z | |
dc.date.available | 2013-04-08T20:50:00Z | |
dc.date.issued | 2009-03 | en_US |
dc.identifier.citation | Foster, David R.; Yee, Shiyin; Bleske, Barry E.; Carver, Peggy L.; Shea, Michael J.; Menon, Sujatha S.; Ramachandran, Chandrasekharan; Welage, Lynda S.; Amidon, Gordon L. (2009). "Lack of Interaction Between the Peptidomimetic Substrates Captopril and Cephradine." The Journal of Clinical Pharmacology 49(3). <http://hdl.handle.net/2027.42/97250> | en_US |
dc.identifier.issn | 0091-2700 | en_US |
dc.identifier.issn | 1552-4604 | en_US |
dc.identifier.uri | https://hdl.handle.net/2027.42/97250 | |
dc.publisher | Blackwell Publishing Ltd | en_US |
dc.publisher | Wiley Periodicals, Inc. | en_US |
dc.subject.other | Cephalosporin | en_US |
dc.subject.other | HPEPT1 | en_US |
dc.subject.other | Drug Interaction | en_US |
dc.subject.other | Peptide Transport | en_US |
dc.subject.other | ACE‐Inhibitor | en_US |
dc.title | Lack of Interaction Between the Peptidomimetic Substrates Captopril and Cephradine | en_US |
dc.type | Article | en_US |
dc.rights.robots | IndexNoFollow | en_US |
dc.subject.hlbsecondlevel | Pharmacy and Pharmacology | en_US |
dc.subject.hlbsecondlevel | Pediatrics | en_US |
dc.subject.hlbtoplevel | Health Sciences | en_US |
dc.description.peerreviewed | Peer Reviewed | en_US |
dc.contributor.affiliationum | Department of Internal Medicine, Medical School, University of Michigan, Ann Arbor, MI | en_US |
dc.contributor.affiliationum | College of Pharmacy, University of Michigan and Department of Pharmacy Services, University Hospital, Ann Arbor, MI | en_US |
dc.contributor.affiliationum | College of Pharmacy, University of Michigan, Ann Arbor, MI | en_US |
dc.contributor.affiliationother | Shiyin Yee Inc., Cupertino, CA | en_US |
dc.contributor.affiliationother | Department of Pharmacy Practice, Purdue University, School of Pharmacy and Pharmaceutical Sciences, Indianapolis, IN | en_US |
dc.contributor.affiliationother | Pfizer, Inc., New London, CT | en_US |
dc.identifier.pmid | 19246733 | en_US |
dc.description.bitstreamurl | http://deepblue.lib.umich.edu/bitstream/2027.42/97250/1/0091270008329554.pdf | |
dc.identifier.doi | 10.1177/0091270008329554 | en_US |
dc.identifier.source | The Journal of Clinical Pharmacology | en_US |
dc.identifier.citedreference | Duchin KL, McKinstry DN, Cohen AI, Migdalof BH. Pharmacokinetics of captopril in healthy subjects and in patients with cardiovascular diseases. Clin Pharmacokinet. 1988; 14: 241 – 259. | en_US |
dc.identifier.citedreference | Lin JH, Chen IW, Ulm EH, Duggan DE. Differential renal handling of angiotensin‐converting enzyme inhibitors enalaprilat and lisinopril in rats. Drug Metab Dispos. 1988; 16: 392 – 396. | en_US |
dc.identifier.citedreference | Yuasa H, Fleisher D, Amidon GL. Noncompetitive inhibition of cephradine uptake by enalapril in rabbit intestinal brush‐border membrane vesicles: an enalapril specific inhibitory binding site on the peptide carrier. J Pharmacol Exp Ther. 1994; 269: 1107 – 1111. | en_US |
dc.identifier.citedreference | Yuasa H, Amidon GL, Fleisher D. Peptide carrier‐mediated transport in intestinal brush border membrane vesicles of rats and rabbits: cephradine uptake and inhibition. Pharm Res. 1993; 10: 400 – 404. | en_US |
dc.identifier.citedreference | Thwaites DT, Hirst BH, Simmons NL. Substrate specificity of the di/tripeptide transporter in human intestinal epithelia (Caco‐2): identification of substrates that undergo H(+)‐coupled absorption. Br J Pharmacol. 1994; 113: 1050 – 1056. | en_US |
dc.identifier.citedreference | Kitagawa S, Takeda J, Sato S. pH‐dependent inhibitory effects of angiotensin‐converting enzyme inhibitors on cefroxadine uptake by rabbit small intestinal brush‐border membrane vesicles and their relationship with hydrophobicity and the ratio of zwitterionic species. Biol Pharm Bull. 1999; 22: 721 – 724. | en_US |
dc.identifier.citedreference | Kitagawa S, Takeda J, Kaseda Y, Sato S. Inhibitory effects of angiotensin‐converting enzyme inhibitor on cefroxadine uptake by rabbit small intestinal brush border membrane vesicles. Biol Pharm Bull. 1997; 20: 449 – 451. | en_US |
dc.identifier.citedreference | Friedman DI, Amidon GL. Intestinal absorption mechanism of dipeptide angiotensin converting enzyme inhibitors of the lysyl‐proline type: lisinopril and SQ 29,852. J Pharm Sci. 1989; 78: 995 – 998. | en_US |
dc.identifier.citedreference | Friedman DI, Amidon GL. Passive and carrier‐mediated intestinal absorption components of two angiotensin converting enzyme (ACE) inhibitor prodrugs in rats: enalapril and fosinopril. Pharm Res. 1989; 6: 1043 – 1047. | en_US |
dc.identifier.citedreference | Matsumoto S, Saito H, Inui K. Transcellular transport of oral cephalosporins in human intestinal epithelial cells, Caco‐2: interaction with dipeptide transport systems in apical and basolateral membranes. J Pharmacol Exp Ther. 1994; 270: 498 – 504. | en_US |
dc.identifier.citedreference | Hu M, Zheng L, Chen J, et al. Mechanisms of transport of quinapril in Caco‐2 cell monolayers: comparison with cephalexin. Pharm Res. 1995; 12: 1120 – 1125. | en_US |
dc.identifier.citedreference | Zhu T, Chen XZ, Steel A, Hediger MA, Smith D. Differential recognition of ACE inhibitors in xenopus laevis oocytes expressing rat PEPT1 and PEPT2. Pharm Res. 2000; 17: 526 – 532. | en_US |
dc.identifier.citedreference | Lukner P, Brandsch M. Interaction of 31 β‐lactum antibiotics with the H+/peptide symporter PEPT2: analysis of affinity constants and comparison with PEPT1. Eur J Pharm Biopharm. 2005; 59: 17 – 24. | en_US |
dc.identifier.citedreference | Moore VA, Irwin WJ, Timmins P, et al. A rapid screening system to determine drug affinities for the intestinal dipeptide transporter 2: affinities of ACE inhibitors. Int J Pharm. 2000; 210: 29 – 44. | en_US |
dc.identifier.citedreference | Bathala MS, Weinstein SH, Meeker FS Jr, Singhvi SM, Migdalof BH. Quantitative determination of captopril in blood and captopril and its disulfide metabolites in plasma by gas chromatography. J Pharm Sci. 1984; 73: 340 – 344. | en_US |
dc.identifier.citedreference | Drummer OH, Jarrot B, Louis WJ. Combined gas chromatographic‐mass spectrometric procedure for the measurement of captopril and sulfur‐conjugated metabolites of captopril in plasma and urine. J Chromatogr. 1984; 305: 83 – 93. | en_US |
dc.identifier.citedreference | Lindgren K. Determination of cefadroxil in serum by highperformance liquid chromatography with cephradine as internal standard. J Chromatogr. 1987; 413: 347 – 350. | en_US |
dc.identifier.citedreference | Gibaldi M, Perrier D. Pharmacokinetics New York: Dekker; 1982: 409 – 417. | en_US |
dc.identifier.citedreference | Nightingale CH, Greene DS, Quintiliani R. Pharmacokinetics and clinical use of cephalosporin antibiotics. J Pharm Sci. 1975; 64: 1899 – 1926. | en_US |
dc.identifier.citedreference | Inui K, Yamamoto M, Saito H. Transepithelial transport of oral cephalosporins by monolayers of intestinal epithelial cell line Caco‐2: specific transport systems in apical and basolateral membranes. J Pharmacol Exp Ther. 1992; 261: 195 – 201. | en_US |
dc.identifier.citedreference | Jacolot A, Tod M, Petitjean O. Pharmacokinetic interaction between cefdinir and two angiotensin‐converting enzyme inhibitors in rats. Antimicrob Agents Chemother. 1996; 40: 979 – 982. | en_US |
dc.identifier.citedreference | Padoin C, Tod M, Perret G, Petitjean O. Analysis of the pharmacokinetic interaction between cephalexin and quinapril by a nonlinear mixed‐effect model. Antimicrob Agents Chemother. 1998; 42: 1463 – 1469. | en_US |
dc.identifier.citedreference | Bins JW, Mattie H. Saturation of the tubular excretion of beta‐lactam antibiotics. Br J Clin Pharmacol. 1988; 25: 41 – 50. | en_US |
dc.identifier.citedreference | van Ginneken CA, Russel FG. Saturable pharmacokinetics in the renal excretion of drugs. Clin Pharmacokinet. 1989; 16: 38 – 54. | en_US |
dc.identifier.citedreference | Landowski CP, Sun D, Foster DR, et al. Gene expression in the human intestine and correlation with oral valacyclovir pharmacokinetic parameters. J Pharmacol Exp Ther. 2003; 306: 778 – 786. | en_US |
dc.identifier.citedreference | Phan DD, Chin‐Hong P, Lin ET, Anderle P, Sadee W, Guglielmo BJ. Intra‐ and interindividual variabilities of valacyclovir oral bioavailability and effect of coadministration of an hPEPT1 inhibitor. Antimicrob Agents Chemother. 2003; 47: 2351 – 2353. | en_US |
dc.identifier.citedreference | Bai JPF, Stewart BH, Amidon GL.: Gastrointestinal transport of peptide and protein drugs and prodrugs. In, Welling PG, Balant LP eds. Handbook of Experimental Pharmacology. Heidelberg: Springer‐Verlag; 1994: 189 – 206. | en_US |
dc.identifier.citedreference | Naruhashi K, Sai Y, Tamai I, Suzuki N, Tsuji A. PepT1 mRNA expression is induced by starvation and its level correlates with absorptive transport of cefadroxil longitudinally in the rat intestine. Pharm Res. 2002; 19: 1417 – 1423. | en_US |
dc.identifier.citedreference | Thamotharan M, Bawani SZ, Zhou X, Adibi SA. Functional and molecular expression of intestinal oligopeptide transporter (Pept‐1) after a brief fast. Metabolism. 1999; 48: 681 – 684. | en_US |
dc.identifier.citedreference | Erickson RH, Gum JR, Lindstrom MM, McKean D, Kim YS. Regional expression and dietary regulation of rat small intestinal peptide and amino acid transporter mRNAs. Biochem Biophys Res Commun. 1995; 216: 249 – 257. | en_US |
dc.identifier.citedreference | Shiraga T, Miyamoto K, Tanaka H, et al. Cellular and molecular mechanisms of dietary regulation on rat intestinal H+/Peptide transporter PepT1. Gastroenterology. 1999; 116: 354 – 362. | en_US |
dc.identifier.citedreference | Adibi SA. Regulation of expression of the intestinal oligopeptide transporter (Pept‐1) in health and disease. Am J Physiol Gastrointest Liver Physiol. 2003; 285: G779 – G788. | en_US |
dc.identifier.citedreference | Thwaites DT, Cavet M, Hirst BH, Simmons NL. Angiotensin‐converting enzyme (ACE) inhibitor transport in human intestinal epithelial (Caco‐ 2) cells. Br J Pharmacol. 1995; 114: 981 – 986. | en_US |
dc.identifier.citedreference | Hu M, Amidon GL. Passive and carrier‐mediated intestinal absorption components of captopril. J Pharm Sci. 1988; 77: 1007 – 1011. | en_US |
dc.identifier.citedreference | Oh D‐M, Han H‐K, Amidon GL.: Drug transport and targeting. In, Amidon GL, Sadee W ed. Membrane Transporters as Drug Targets. New York, NY: Klewer Academis/Plenum; 1999: 59 – 88. | en_US |
dc.identifier.citedreference | Eberl S, Renner B, Neubert A, et al. Role of p‐glycoprotein inhibition for drug interactions:Evidence from in vitro and pharmacoepidemiological studies. Clin Pharmacokinet. 2007; 46: 1039 – 1049. | en_US |
dc.identifier.citedreference | Callaghan R, Crowley E, Potter S, Kerr ID. P‐glycoprotein: so many ways to turn it on. J Clin Pharmacol. 2008; 48: 365 – 378. | en_US |
dc.identifier.citedreference | Tsuji A, Tamai I. Carrier‐mediated intestinal transport of drugs. Pharm Res. 1996; 13: 963 – 977. | en_US |
dc.identifier.citedreference | Sai Y. Biochemical and molecular pharmacological aspects of transporters as determinants of drug disposition. Drug Metab Pharmacokinet. 2005; 20: 91 – 99. | en_US |
dc.identifier.citedreference | Herrera‐Ruiz D, Knipp GT. Current perspectives on established and putative mammalian oligopeptide transporters. J Pharm Sci. 2003; 92: 691 – 714. | en_US |
dc.identifier.citedreference | Brodin B, Ielsen CU, Teffansen B, Fokjaer S. Transport of peptidomimetic drugs by the intestinal Di/tri‐peptide transporter, PepT1. Pharmacol Toxicol. 2002; 90: 285 – 296. | en_US |
dc.identifier.citedreference | Terada T, Inui KI. Peptide transporters: structure, function, regulation and application for drug delivery. Curr Drug Metab. 2004; 5: 85 – 94. | en_US |
dc.identifier.citedreference | Anand BS, Patel J, Mitra AK. Interactions of the dipeptide ester prodrugs of acyclovir with the intestinal oligopeptide transporter: competitive inhibition of glycylsarcosine transport in human intestinal cell line‐caco‐2. J Pharmacol. 2003; 2: 781 – 791. | en_US |
dc.identifier.citedreference | Irie M, Terada T, Sawada K, Saito H, Inui KI. Recognition and transport characteristics of nonpeptidic compounds by basolateral peptide transporter in caco‐2 cells. J Pharmacol. 2001; 298: 711 – 717. | en_US |
dc.identifier.citedreference | Lepsy CS, Guttendorf RJ, Kugler AR, Smith DE. Effects of organic anion, organic cation, and dipeptide transport inhibitors on cefdinir in the isolated perfused rat kidney. Antimicrob Agents Chemother. 2003; 47: 689 – 696. | en_US |
dc.identifier.citedreference | Berger UV, Hediger MA. Distribution of peptide transporter PEPT2 mRNA in the rat nervous system. Anat Embryol (Berl). 1999; 199: 439 – 449. | en_US |
dc.identifier.citedreference | Bahadduri PM, D'Souza VM, Pinsonneault JK, et al. Functional characterization of the peptide transporter PEPT2 in primary cultures of human upper airway epithelium. Am J Respir Cell Mol Biol. 2005; 32: 319 – 325. | en_US |
dc.identifier.citedreference | Shu C, Shen H, Hopfer, U, Smith DE. Mechanism of intestinal absorption and renal reabsorption of an orally active ace inhibitor: uptake and transport of fosinopril in cell cultures. Drug Metab Dispos. 2001; 29: 1307 – 1315. | en_US |
dc.identifier.citedreference | Lin CJ, Smith DE. Glycylsarcosine uptake in rabbit renal brush border membrane vesicles isolated from outer cortex or outer medulla: evidence for heterogeneous distribution of oligopeptide transporters. AAPS Pharm Sci. 1999; 1: E1. | en_US |
dc.owningcollname | Interdisciplinary and Peer-Reviewed |
Files in this item
Remediation of Harmful Language
The University of Michigan Library aims to describe library materials in a way that respects the people and communities who create, use, and are represented in our collections. Report harmful or offensive language in catalog records, finding aids, or elsewhere in our collections anonymously through our metadata feedback form. More information at Remediation of Harmful Language.
Accessibility
If you are unable to use this file in its current format, please select the Contact Us link and we can modify it to make it more accessible to you.