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Pyrimido[4,5‐ d ]pyrimidin‐4(1 H )‐one Derivatives as Selective Inhibitors of EGFR Threonine 790 to Methionine 790 (T790M) Mutants
dc.contributor.authorXu, Tianfengen_US
dc.contributor.authorZhang, Lianwenen_US
dc.contributor.authorXu, Shilinen_US
dc.contributor.authorYang, Chao‐yieen_US
dc.contributor.authorLuo, Jinfengen_US
dc.contributor.authorDing, Fangen_US
dc.contributor.authorLu, Xiaoyunen_US
dc.contributor.authorLiu, Yingxueen_US
dc.contributor.authorTu, Zhengchaoen_US
dc.contributor.authorLi, Shiliangen_US
dc.contributor.authorPei, Duanqingen_US
dc.contributor.authorCai, Qianen_US
dc.contributor.authorLi, Honglinen_US
dc.contributor.authorRen, Xiaomeien_US
dc.contributor.authorWang, Shaomengen_US
dc.contributor.authorDing, Keen_US
dc.date.accessioned2013-09-04T17:18:41Z
dc.date.available2014-10-06T19:17:42Zen_US
dc.date.issued2013-08-05en_US
dc.identifier.citationXu, Tianfeng; Zhang, Lianwen; Xu, Shilin; Yang, Chao‐yie ; Luo, Jinfeng; Ding, Fang; Lu, Xiaoyun; Liu, Yingxue; Tu, Zhengchao; Li, Shiliang; Pei, Duanqing; Cai, Qian; Li, Honglin; Ren, Xiaomei; Wang, Shaomeng; Ding, Ke (2013). "Pyrimido[4,5â d ]pyrimidinâ 4(1 H )â one Derivatives as Selective Inhibitors of EGFR Threonine 790 to Methionine 790 (T790M) Mutants ." Angewandte Chemie International Edition 52(32): 8387-8390. <http://hdl.handle.net/2027.42/99681>en_US
dc.identifier.issn1433-7851en_US
dc.identifier.issn1521-3773en_US
dc.identifier.urihttps://hdl.handle.net/2027.42/99681
dc.publisherWILEY‐VCH Verlagen_US
dc.subject.otherInhibitorsen_US
dc.subject.otherT790M Mutantsen_US
dc.subject.otherSelectivityen_US
dc.subject.otherDrug Designen_US
dc.titlePyrimido[4,5‐ d ]pyrimidin‐4(1 H )‐one Derivatives as Selective Inhibitors of EGFR Threonine 790 to Methionine 790 (T790M) Mutantsen_US
dc.typeArticleen_US
dc.rights.robotsIndexNoFollowen_US
dc.subject.hlbsecondlevelChemistryen_US
dc.subject.hlbtoplevelScienceen_US
dc.description.peerreviewedPeer Revieweden_US
dc.contributor.affiliationumThe University of Michigan Comprehensive Cancer Center, Ann Arbor, MI 48109 (USA)en_US
dc.contributor.affiliationotherInstitute of Chemical Biology, Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences, 190 Kaiyuan Avenue, Guangzhou 510530 (China)en_US
dc.contributor.affiliationotherUniversity of Chinese Academy of Sciences, 19 Yuquan Road, Beijing 100049 (China)en_US
dc.contributor.affiliationotherEast China University of Science and Technology, 130 Meilong Road, Shanghai 200237 (China)en_US
dc.contributor.affiliationotherInstitute of Chemical Biology, Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences, 190 Kaiyuan Avenue, Guangzhou 510530 (China)en_US
dc.identifier.pmid23804305en_US
dc.description.bitstreamurlhttp://deepblue.lib.umich.edu/bitstream/2027.42/99681/1/8387_ftp.pdf
dc.description.bitstreamurlhttp://deepblue.lib.umich.edu/bitstream/2027.42/99681/2/anie_201302313_sm_miscellaneous_information.pdf
dc.identifier.doi10.1002/anie.201302313en_US
dc.identifier.sourceAngewandte Chemie International Editionen_US
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dc.owningcollnameInterdisciplinary and Peer-Reviewed


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